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CBP73XXXX kinase 激酶稳定细胞株

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品牌 自营品牌 供货周期 两周

激酶(kinase)是一类从高能供体分子(如ATP)转移磷酸基团到特定靶分子(底物)的酶;这一过程谓之磷酸化许多肿瘤的发生是由某些与生长相关的“激酶”发生突变导致异常活化引起的,因而针对这些突变激酶的YZ剂能够有效YZ这些激酶的活性,从而达到YZ癌细胞增长的目的。

产品优势

a. 基因变化背景单一可控,细胞生存依赖*转基因导入的活化激酶不存在脱靶现象,能够更加准确快速地表明药物的作用机制。

b. 结合高通量药物筛选平台,实现了批量化合物JZ靶点检测与选择性评价,检测药物的靶点选择性,评价药物毒副反应。

 

现货细胞列表(更多产品请咨询客服4008750250)

kinase targetcell linesCat.NO
ABL (BCR-ABL)Ba/F3/ABL (BCR-ABL)CBP73001
ACVR1B/BMPR2U2OS/ACVR1B/BMPR2CBP73002
ACVR1C/ACVR2U2OS/ACVR1C/ACVR2CBP73003
ACVR1C/ACVR2BU2OS/ACVR1C/ACVR2BCBP73004
ACVR2/ACVR1U2OS/ACVR1/ACVR2 CBP73005
ACVRL1/ACVR2U2OS/ACVRL1/ACVR2 CBP73006
ACVRL1/ACVR2BU2OS/ACVRL1/ACVR2BCBP73007
ACVRL1/BMPR2U2OS/ACVRL1/BMPR2CBP73008
ALKBa/F3/ALKCBP73009
ARG (ABL2)Ba/F3/ARG (ABL2)CBP73010
AXLU2OS/AXLCBP73011
BLKU2OS/BLK CBP73012
BLKHEK293/BLK CBP73013
BMPR1A/ACVR2U2OS/BMPR1A/ACVR2ACBP73014
BMPR1A/ACVR2BU2OS/BMPR1A/ACVR2BCBP73015
BMPR1A/ACVR2BU2OS/BMPR1A/ACVR2B CBP73016
BMPR1A/BMPR2U2OS/BMPR1A/BMPR2CBP73017
BMPR1A/BMPR2U2OS/BMPR1A/BMPR2CBP73018
BMPR1B/ACVR2U2OS/BMPR1B/ACVR2ACBP73019
BMPR1B/ACVR2U2OS/BMPR1B/ACVR2ACBP73020
BMPR1B/ACVR2BU2OS/BMPR1B/ACVR2BCBP73021
BMPR1B/BMPR2U2OS/BMPR1B/BMPR2CBP73022
BMXBa/F3/BMXCBP73023
BTKA549/BTKCBP73024
CCK4 (PTK7)Ba/F3/CCK4 (PTK7)CBP73025
cINSRaU2OS/cINSRa CBP73026
cINSRbU2OS/cINSRb CBP73027
c-KITU2OS/c-KITCBP73028
CLK1HEK293/CLK1 CBP73029
CLK2 A549/CLK2CBP73030
c-MET/c-METU2OS/c-MET/c-METCBP73031
c-Ret-GFRα1U2OS/c-Ret-GFRα1CBP73032
c-Ret-GFRα2U2OS/c-Ret-GFRα2CBP73033
CSF1RA549/CSF1RCBP73034
CSF1R/CSF1RU2OS/CSF1R/CSF1RCBP73035
CSF3R-JAK1U2OS/CSF3R-JAK1CBP73036
CSNK1DA549/CSNK1DCBP73037
DDR1U2OS/DDR1CBP73038
DDR2Ba/F3/DDR2CBP73039
EGFR [L858R]Ba/F3/EGFR [L858R]CBP73040
EGFR [T790M]Ba/F3/EGFR [T790M]CBP73041
EGFR/EGFRU2OS/EGFR/EGFRCBP73042
EGFR/ErbB2U2OS/EGFR/ErbB2CBP73043
EGFR/ErbB3U2OS/EGFR/ErbB3CBP73044
EGFR[D746-750]Ba/F3/EGFR[D746-750]CBP73045
EGFR[D746-750+T790M]Ba/F3/EGFR[D746-750+T790M]CBP73046
EGFR[L858R+C797S] Ba/F3/EGFR[L858R+C797S] CBP73047
EGFR[L858R+T790M]Ba/F3/EGFR[L858R+T790M]CBP73048
EGFR[L858R+T790M+C797S]Ba/F3/EGFR[L858R+T790M+C797S]CBP73049
EGFR[L861Q] Ba/F3/EGFR[L861Q] CBP73050
EGFR[L861Q+T790M]Ba/F3/EGFR[L861Q+T790M]CBP73051
EGFR[L861Q+T790M]Ba/F3/EGFR[L861Q+T790M]CBP73052
EphA1Ba/F3/EphA1CBP73053
EphA3Ba/F3/EphA3CBP73054
EphA4U2OS/EphA4CBP73055
EphA5U2OS/EphA5CBP73056
EphA7U2OS/EphA7CBP73057
EphB1U2OS/EphB1CBP73058
EphB2U2OS/EphB2CBP73059
EphB3U2OS/EphB3CBP73060
EphB4U2OS/EphB4CBP73061
EpoR-JAK2U2OS/EpoR-JAK2CBP73062
ErbB1U2OS/ErbB1CBP73063
ErbB2/ErbB3U2OS/ErbB2/ErbB3CBP73064
ErbB2/ErbB4U2OS/ErbB2/ErbB4CBP73065
ErbB2-ErbB3U2OS/ErbB2-ErbB3CBP73066
ErbB4U2OS/ErbB4CBP73067
ErbB4/ErbB4U2OS/ErbB4/ErbB4CBP73068
FAKBa/F3/FAKCBP73069
FGFR1U2OS/FGFR1CBP73070
FGFR1 [V561M]Ba/F3/FGFR1 [V561M]CBP73071
FGFR1-α-KlothoU2OS/FGFR1-α-KlothoCBP73072
FGFR1-β-KlothoU2OS/FGFR1-β-KlothoCBP73073
FGFR1-β-KlothoU2OS/FGFR1-β-KlothoCBP73074
FGFR2U2OS/FGFR2CBP73075
FGFR2 [K660E]Ba/F3/FGFR2 [K660E]CBP73076
FGFR2 [K660N]Ba/F3/FGFR2 [K660N]CBP73077
FGFR2 [N550K]Ba/F3/FGFR2 [N550K]CBP73078
FGFR2 [V565I]Ba/F3/FGFR2 [V565I]CBP73079
FGFR2/AFF3Ba/F3/FGFR2/AFF3CBP73080
FGFR2/BICC1 Ba/F3/FGFR2/BICC1 CBP73081
FGFR2/CASP7Ba/F3/FGFR2/CASP7CBP73082
FGFR2/CCDC6Ba/F3/FGFR2/CCDC6CBP73083
FGFR3Ba/F3/FGFR3CBP73084
FGFR3 [K650M]Ba/F3/FGFR3 [K650M]CBP73085
FGFR3(G380R)/FGFR3(G380R)U2OS/FGFR3(G380R)/FGFR3(G380R)CBP73086
FGFR3/BAIAP2LBa/F3/FGFR3/BAIAP2LCBP73087
FGFR3/FGFR3U2OS/FGFR3/FGFR3CBP73088
FGFR4U2OS/FGFR4CBP73089
FGFR4 [V550E]Ba/F3/FGFR4 [V550E]CBP73090
FGFR4-α-KlothoU2OS/FGFR4-α-KlothoCBP73091
FGFR4-β-KlothoU2OS/FGFR4-β-KlothoCBP73092
FGRHEK293/FGRCBP73093
FLT1(VEGFR1)Ba/F3/FLT1(VEGFR1)CBP73094
FLT3U2OS/FLT3CBP73095
FLT3-ITDBa/F3/FLT3-ITDCBP73096
FLT3-ITD [D835V]Ba/F3/FLT3-ITD [D835V]CBP73097
FLT3-ITD [D835Y] Ba/F3/FLT3-ITD [D835Y] CBP73098
FLT3-ITD [F691L]Ba/F3/FLT3-ITD [F691L] CBP73099
FLT3-ITD [Y842C]Ba/F3/FLT3-ITD [Y842C]CBP73100
FLT3-ITD [Y842H]Ba/F3/FLT3-ITD [Y842H]CBP73101
FLT4U2OS/FLT4CBP73102
FLT4(VEGFR3)Ba/F3/FLT4(VEGFR3)CBP73103
FMS (CSF1R)Ba/F3/FMS (CSF1R)CBP73104
FRKBa/F3/FRKCBP73105
FYNBa/F3/FYNCBP73106
GHR-JAK1U2OS/GHR-JAK1CBP73107
GHR-JAK2U2OS/GHR-JAK2CBP73108
HCKA549/HCKCBP73109
HER2(ERBB2)Ba/F3/HER2(ERBB2)CBP73110
HER3 (ERBB3)Ba/F3/HER3 (ERBB3)CBP73111
IGF1RHEK293/IGF1RCBP73112
INSRBa/F3/INSRCBP73113
INSRaU2OS/INSRaCBP73114
INSRbU2OS/INSRbCBP73115
JAK1Ba/F3/JAK1CBP73116
JAK2Ba/F3/JAK2CBP73117
JAK3U2OS/JAK3CBP73118
KDRU2OS/KDRCBP73119
KDR(VEGFR2)Ba/F3/KDR(VEGFR2)CBP73120
KDR/KDRHEK293/KDR/KDRCBP73121
LCKU2OS/LCKCBP73122
LYNBa/F3/LYNCBP73123
MEK1A549/MEK1CBP73124
MER (MERTK)Ba/F3/MER (MERTK)CBP73125
METBa/F3/METCBP73126
mINSRaU2OS/mINSRaCBP73127
mINSRbU2OS/mINSRbCBP73128
PDGFRaU2OS/PDGFRaCBP73129
PDGFRbU2OS/PDGFRbCBP73130
PI3KδHEK293/PI3KδCBP73131
PIM1A549/PIM1CBP73132
PLCG1(SH2)-EAU2OS/PLCG1-EACBP73133
PRLR-JAK1U2OS/PRLR-JAK1CBP73134
PRLR-JAK2U2OS/PRLR-JAK2CBP73135
PYK2A549/PYK2CBP73136
RETBa/F3/RETCBP73137
RET [V804M]Ba/F3/RET [V804M]CBP73138
rhTrkA-rhP75U2OS/rhTrkA-rhP75CBP73139
RIPK1Jurkat/RIPK1CBP73140
RIPK2HEK293/RIPK2CBP73141
RIPK3Jurkat/RIPK3CBP73142
RON (MST1R)Ba/F3/RON (MST1R)CBP73143
ROR1Ba/F3/ROR1CBP73144
rTrkA-rP75U2OS/rTrkA-rP75CBP73145
RYKBa/F3/RYKCBP73146
SHC1(SH2)-EAU2OS/SHC1-EACBP73147
SIK1A549/SIK1CBP73148
SRCBa/F3/SRCCBP73149
SYKBa/F3/SYKCBP73150
SYKU2OS/SYKCBP73151
TGFBR1/TGFBR2U2OS/TGFBR1/TGFBR2CBP73152
TGFBR1/TGFBR2/ENGU2OS/TGFBR1/TGFBR2/ENGCBP73153
TIE1Ba/F3/TIE1CBP73154
TIE2HEK293/TIE2CBP73155
TRKA (NTRK1)Ba/F3/TRKA (NTRK1)CBP73156
TrkA-P75U2OS/TrkA-P75CBP73157
TRKB (NTRK2)Ba/F3/TRKB (NTRK2)CBP73158
TrkB-P75U2OS/TrkB-P75CBP73159
TRKC (NTRK3)Ba/F3/TRKC (NTRK3)CBP73160
TrkC-P75U2OS/TrkC-P75CBP73161
TYK2U2OS/TYK2CBP73162
TYRO3U2OS/TYRO3CBP73163
YES1U2OS/YES1CBP73164
ZAP70Ba/F3/ZAP70CBP73165

 

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