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BCl-2 Inhibitor, ABT-199

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BCl-2 Inhibitor, ABT-199
Product Name: BCl-2 Inhibitor, ABT-199
Alternate Name/Synonyms: 2-((1H-Pyrrolo[2,3-b]pyridin-5-yl)oxy)-4-(4-((4’-chloro-5,5-dimethyl-3,4,5,6-tetrahydro-[1,1’-biphenyl]-2-yl)methyl)piperazin-1-yl)-N-((3-nitro-4-(((tetrahydro-2H-pyran-4-yl)methyl)amino)phenyl)sulfonyl)benzamide; GDC-0199
Description: Cell-permeable. A potent and selective BCl-2 inhibitor that spares platelets while achieving potent antitumor activity.
Peptide Sequence: N/A
Appearance: White to off-white solid
Formulation: N/A
CAS Number: 1257044-40-8
Molecular Formula: C45H50ClN7O7S
Molecular Weight: 868.44
Purity: ≥98% by HPLC
Solubility: DMSO (50 mM)
Storage Temp.: -20°C
Shipping Conditions: gel pack Protect from light and moisture
Handling:
USAGE: For Research Use Only! Not For Use in Humans
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