Pyrazolylpyrrole ERK Inhibitor,N-[1-(3-chloro-4-fluorophenyl)-2-hydroxyethyl]-4-[4-(3-chlorophenyl)-1,2-dihydropyrazol-3-ylidene]pyrrole-2-carboxamide,933786-58-4

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产品名称：Pyrazolylpyrrole ERK Inhibitor

产品别名：N-[1-(3-chloro-4-fluorophenyl)-2-hydroxyethyl]-4-[4-(3-chlorophenyl)-1,2-dihydropyrazol-3-ylidene]pyrrole-2-carboxamide

CAS号：933786-58-4

英文别名：N-[1-(3-chloro-4-fluorophenyl)-2-hydroxyethyl]-4-[4-(3-chlorophenyl)-1,2-dihydropyrazol-3-ylidene]pyrrole-2-carboxamide

分子量：459.3

分子式：C₂₂H₁₇Cl₂FN₄O₂

纯度：>98%

外观：见爱必信官网

保存方法：Store at -20° C

描述：Pyrazolylpyrrole ERK Inhibitor is a potent, ATP-competitive inhibitor of ERK2 (K_i = 2 nM). This compound is highly selective for ERK2 compared to other kinases such as PKA (K_i = 0.39 µM) and JNK3 (K_i = 4 µM). Inhibits proliferation of Colo205 cells with an IC₅₀ value of 0.54 µM.

应用：A potent inhibitor of ERK2

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