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Glucagon Receptor Antagonist, Control,Glucagon Receptor Antagonist, Control,362482-00-6

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    试剂描述:

    产品名称:Glucagon Receptor Antagonist, Control

    产品别名:N-(3-Cyano-6-(1,1-dimethylpropyl)-4,5,6,7-tetrahydro-1-benzothien-2-yl)-4-bromobenzamide

    CAS号:362482-00-6

    英文别名:N-(3-Cyano-6-(1,1-dimethylpropyl)-4,5,6,7-tetrahydro-1-benzothien-2-yl)-4-bromobenzamide

    分子量:431.4

    分子式:C21H23BrN2OS

    纯度:见爱必信官网

    外观:见爱必信官网

    保存方法:Store at 4° C

    描述:Glucagon Receptor Antagonist, Control is a cell-permeable thienyl-amide compound that serves as an inactive control for Glucagon Receptor Antagonist. Glucagon Receptor Antagonist, Control displays weak affinity for hGCGR and is ineffective when preventing glucagon binding (20% inhibition at 10 μM in membranes prepared from CHO-hGCGR) and glucagon-, forskolin-, and GIP-induced cAMP production (10% inhibition in CHO-hGCGR cells). Only minimally suppresses glucagon-induced glycogenolysis in human primary hepatocytes.

    应用:A compound that serves as an inactive control for Glucagon Receptor Antagonist

    产品信息订购:

      产品货号   产品名称   规格 价格 大包装及货期
      abs42019041   Glucagon Receptor Antagonist, Control   1mg  2340   立即咨询

    产品更多信息请进入爱必信网站咨询

    温馨提示:不可用于临床ZL。
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