Solcitinib,1206163-45-2

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YZ剂描述：

产品名称：Solcitinib

产品别名：(GLPG0778,GSK2586184)

英文别名：GLPG 0778;GSK 2586184;GLPG-0778;GSK-2586184

靶点：JAK1

CAS：1206163-45-2

纯度：＞98%

外观：Powder

保存方法：store at -20℃ for one year（Powder）； in DMSO or others solvent store at 2-4℃ for two weeks, at -20℃ for six months.

描述：

Solcitinib, also known as GSK2586184 or GLPG0778, is a Janus kinase 1 (JAK1) inhibitor.

溶解性：DMSO : 20 mg/mL (51.35 mM; Need ultrasonic and warming)

体外研究：

Solcitinib is an orally active, competitive, potent, selective JAK1 inhibitor, with an IC50 of 9.8 nM, and 11-, 55- and 23-fold selectivity over JAK2, JAK3 and TYK2, respectively. Solcitinib is used in the research of moderate-to-severe plaque-type psoriasis.

体内研究：

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