产品:4-Desfluoro-6-fluoro Dolutegravir 分子式:C20H19F2N3O5 分子量:419.38 性状外观:No Data Available 溶点:No Data Available 溶解性:No Data Available
4-Desfluoro-6-fluoro Dolutegravir is impurity C of Dolutegravir (D528800), which is a second generation HIV-1 integrase strand transfer inhibitor. Dolutegravir is currently in Phase III clinical trials for the treatment of HIV infection. Dolutegravir has been shown to potently inhibit HIV replication in cells such as peripheral blood mononuclear cells (PBMCs), MT-4 cells and CIP4 cells infected with a self-inactivating PHIV lentiviral vector.