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Acetyl-(Cys¹¹,D-2-Nal¹⁴,Cys¹⁸)-β-MSH (11-22) amide trifluoroacetate salt

产品信息
  • 规格:1mg产品价格:5250.00
    规格:5mg产品价格:21015.00
    Catalog Number H-4352
    Synonyms HS014
    Molecular Formula C₇₁H₉₄N₂₀O₁₇S₂
    Relative Molecular Mass 1563.78
    CAS Registry Number [207678-81-7] net
    Source Synthetic
    Storage Conditions -20 ± 5 °C
    Areas of Interest Obesity Research|Pituitary & Hypothalamic Hormones
    产品描述
    The cyclic MSH analog HS014, which has potent and highly selective antagonistic activity at the MC4 receptor in vitro, strongly stimulates food intake in satiated rats. Therefore, HS014 appears to be a useful tool to investigate the physiology of the MC4 receptor.
    论文引用
    • B.L.Panaro et al., Cell Metab., 20, 1018 (2014)
    • L.Zvejniece et al., Pharmacol. Biochem. Behav., 85, 287 (2006)
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